Metabotropic glutamate receptor 5 (mGluR5)

Order number PP106-0
Name FPEB
Chemical Formula C14H7FN2
Molecular Weight 222.22
Purity >95%
Packaging min. 10 mg, or as ordered
Purpose Reference standard for [18F]FPEB
Other name 3-Fluoro-5-(pyridinylethynyl)benzonitrile
CA index name Benzonitrile, 3-fluoro-5-[2-(2-pyridinyl)ethynyl]-
Literature Dean F. Wong, Rikki Waterhouse, Hiroto Kuwabara, Jongho Kim, James R. Brašić, Wichana Chamroonrat, Michael Stabins, Daniel P. Holt, Robert F. Dannals, Terence G. Hamill and P. David Mozley. Journal of Nuclear Medicine, March 2013, 54 (3), 388-396.
DOI: https://doi.org/10.2967/jnumed.112.107995
Dupont, AC., Serrière, S., Barantin, L. et al. Study of influence of the glutamatergic concentration of [18F]FPEB binding to metabotropic glutamate receptor subtype 5 with N-acetylcysteine challenge in rats and SRM/PET study in human healthy volunteers. Transl Psychiatry 11, 66 (2021). https://doi.org/10.1038/s41398-020-01152-2