Dopamine

Order number PP006-0
Name FLB 457
Chemical Formula C16H23BrN2O3・HBr
Molecular Weight 452.19
Purity > 95%
Packaging min. 10 mg, or as ordered
Purpose Reference standard for [11C]FLB 457
Other name (S)-(-)-5-Bromo-2,3-dimethoxy N-[(1-ethyl-2-pyrrolidinyl)methyl]benzamide
CA index name Benzamide, 5-bromo-N-[[(2S)-1-ethyl-2-pyrrolidinyl]methyl]-2,3-dimethoxy-
Literature 1. Halldin C, Farde L, Högberg T, Mohell N, Hall H, Suhara T, Karlsson P, Nakashima Y, Swahn CG. Carbon-11-FLB 457: a radioligand for extrastriatal D2 dopamine receptors. J Nucl Med. 1995;36(7):1275-81.
2. Farde L, Suhara T, Nyberg S, Karlsson P, Nakashima Y, Hietala J, Halldin C. A PET-study of [11C]FLB 457 binding to extrastriatal D2-dopamine receptors in healthy subjects and antipsychotic drug-treated patients. Psychopharmacology (Berl). 1997;133(4):396-404.
3. Okubo Y, Olsson H, Ito H, Lofti M, Suhara T, Halldin C, Farde L. PET mapping of extrastriatal D2-like dopamine receptors in the human brain using an anatomic standardization technique and [11C]FLB 457. Neuroimage. 1999;10(6):666-74.
  Selective D2 Receptor Antagonist